Basic Peptide Information

DICL ID
DICL_Pep_02460
Ion Channel
Sodium channel type 8 subunit alpha
Peptide Function
Inhibitor
Gene Name
Scn8a

Activity Data (nM)

IC50
547 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
MKVTLIAILTCAALLVLLHTTAAEELEAQEESQLMEVGMPDTELAALDEERIFECSISCEIEKEGNGKKCKPKKCKGGWKCKFNICVKV
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
μ-TrtX-Ca1a
Peptide Species
C. albostriatus
Peptide Name
Not available
CAS Number
Not available

Experimental Conditions

pH
pH 7.4
Holding Potential (mV)
–110 to -10 mV
Temperature
20–25 °C
Test Method
Patch-clamping
Test Species
Not specified

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available